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公司新闻
免疫检查点活性蛋白及相关产品 CTLA-4,PD-1,IDO1,B7-H4,LAG-3,Tim-3
发布时间:2023-11-16 08:52 | 点击次数:199
免疫检查点活性蛋白及相关产品
CTLA-4,PD-1,IDO1,B7-H4,LAG-3,Tim-3
◆活性免疫检测点蛋白
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B7-H4 (human):Fc (human) (rec.)
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CHI-HF-210B7H4
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B7-H4 (mouse):Fc (mouse) (rec.)
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CHI-MF-110B7H4
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CTLA-4 (human):Fc (human) (rec.)
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CHI-HF-210A4
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CTLA-4 (human):Fc (human) (rec.) (non-lytic)
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CHI-HF-220A4
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CTLA-4 (human):Fc (mouse) (rec.)
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CHI-HF-211A4
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CTLA-4 (mouse):Fc (mouse) (rec.)
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CHI-MF-110A4
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CTLA-4 (mouse):Fc (mouse) (rec.) (non-lytic)
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CHI-MF-120A4
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PD-1 (human):Fc (human) (rec.)
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CHI-HF-210PD1
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PD-1 (human):Fc (human) (rec.) (non-lytic)
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CHI-HF-220PD1
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PD-1 (mouse):Fc (mouse) (rec.)
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CHI-MF-110PD1
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PD-L1/B7-H1 (human):Fc (human) (rec.)
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CHI-HF-210PDL1
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PD-L1/B7-H1 (human):Fc (human) (rec.) (non-lytic)
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CHI-HF-220PDL1
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PD-L1/B7-H1 (mouse):Fc (mouse) (rec.)
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CHI-MF-110PDL1
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PD-L1/B7-H1 (mouse):Fc (mouse) (rec.) (non-lytic)
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CHI-MF-120PDL1
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PD-L2 (human):Fc (human) (rec.)
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CHI-HF-210PDL2
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PD-L2 (human):Fc (human) (rec.) (non-lytic)
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CHI-HF-220PDL2
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PD-L2 (mouse):Fc (mouse) (rec.)
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CHI-MF-110PDL2
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◆IDO1酶&主要抑制剂
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IDO1 (human) Enzyme+Inhibitor Set
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AG-44B-0006
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IDO1 (human) (rec.) (His) (highly active)
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AG-40B-0161
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MMG-0358 Potent Triazole IDO1 Inhibitor AG-CR1-3630
IC50值,mIDO1细胞检测是2 nM,hIDO1细胞检测是80 nM,hIDO1(pH 6.5)酶活检测是330 nM,hIDO1(pH7.4)的酶活检测是71 nM。体内有活性。
参考文献
Rational design of 4-aryl-1,2,3-triazoles for indoleamine 2,3-dioxygenase 1 inhibition: U.F. Roehrig, et al.; J. Med. Chem. , 55, 5270 (2012)
◆肿瘤免疫治疗的LAG-3
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功能性封闭抗体
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LAG-3 (human), mAb (blocking) (17B4)
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AG-20B-0012
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LAG-3 (human), mAb (blocking) (17B4) (preservative free)
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AG-20B-0012PF
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LAG-3, mAb (blocking) (11E3)
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AG-20B-0011
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LAG-3, mAb (blocking) (11E3) (preservative free)
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AG-20B-0011PF
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生物活性蛋白
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LAG-3 (human):Fc (human) (rec.)
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AG-40B-0031
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LAG-3 (mouse):Fc (mouse) (rec.)
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AG-40B-0039
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◆T-细胞免疫球蛋白和粘蛋白结构域
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Tim-3 (human):Fc (human) (rec.)
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CHI-HF-210T3
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Tim-3 (mouse):Fc (mouse) (rec.)
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CHI-MF-110T3
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◆CD1d配体抗肿瘤佐剂
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α-Galactosylceramide
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Potent NKT Cell stimulator
强有效NKT 激活剂
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AG-CN2-0013
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在人类和小鼠NKT细胞里MHC-I蛋白和CD1d分子脂质结合的特异性配体。
参考文献
LIT: Combination of the toll like receptor agonist and α-Galactosylceramide as an efficient adjuvant for cancer vaccine: F. Gableh, et al.; J. Biomed. Sci., 23, 16 (2016)
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